Publications

Publications @ University of Vienna

2025

Kronberger J, Balber T, Schueffl H, Wahrmann R, Federa A, Gradl M et al. Site-Selectively Functionalized Albumin with DFO*Maleimide for ⁸⁹Zr-Radiolabeling Yields a Metabolically Stable PET Probe that Enables Late Time-Point Tumor Imaging in Mice. Journal of Medicinal Chemistry. 2025 Jun 26;68(12):12925-12939. doi: 10.1021/acs.jmedchem.5c00803

Feiner IVJ, Svatunek D, Pressler M, Demuth T, Guarrochena X, Sterba JH et al. Towards DFO*¹²—Preliminary Results of a New Chelator for the Complexation of Actinium-225. Pharmaceutics. 2025 Mar;17(3):320. doi: 10.3390/pharmaceutics17030320

Guarrochena X, Anderla M, Salomon P, Feiner IVJ, Nock BA, Maina T et al. Combination of the amide-to-triazole substitution strategy with alternative structural modifications for the metabolic stabilization of tumor-targeting, radiolabeled peptides. Journal of Peptide Science. 2025 Jan;31(1):e3654. doi: 10.1002/psc.3654

Federa A, Schueffl H, Minichmayr IK, Kastner A, Kronberger J, Mindt TL et al. Comparative Evaluation of Thiol- and Amine-Conjugating Moieties for Endogenous Albumin Binding after Intravenous Administration. ACS Pharmacology and Translational Science. 2025. Epub 2025. doi: 10.1021/acsptsci.5c00240

2024

Guarrochena X, Kanellopoulos P, Stingeder A, Rečnik LM, Feiner IVJ, Brandt M et al. Amide-to-Triazole Switch in Somatostatin-14-Based Radioligands: Impact on Receptor Affinity and In Vivo Stability. Pharmaceutics. 2024 Mar;16(3):392. doi: 10.3390/pharmaceutics16030392

Guarrochena X, Kronberger J, Tieber M, Ciesielski P, Mindt TL, Feiner IVJ. Straightforward Synthesis of DFO* - An Octadentate Chelator for Zirconium-89. ChemMedChem. 2024 Feb 1;19(3):e202300495. doi: 10.1002/cmdc.202300495

Happl B, Balber T, Heffeter P, Denk C, Welch JM, Köster U et al. Synthesis and preclinical evaluation of BOLD-100 radiolabeled with ruthenium-97 and ruthenium-103. Dalton Transactions. 2024. Epub 2024. doi: 10.1039/d4dt00118d

2023

Schmitl S, Raitanen J, Witoszynskyj S, Patronas EM, Nics L, Ozenil M et al. Quality Assurance Investigations and Impurity Characterization during Upscaling of [¹⁷⁷Lu]Lu-PSMA^I&T. Molecules. 2023 Dec;28(23):7696. doi: 10.3390/molecules28237696

Happl B, Brandt M, Balber T, Benčurová K, Talip Z, Voegele A et al. Synthesis and Preclinical Evaluation of Radiolabeled [¹⁰³Ru]BOLD-100. Pharmaceutics. 2023 Nov;15(11):2626. doi: 10.3390/pharmaceutics15112626

Wang Y, Felder PS, Mesdom P, Blacque O, Mindt TL, Cariou K et al. Towards Ruthenium(II)-Rhenium(I) Binuclear Complexes as Photosensitizers for Photodynamic Therapy. ChemBioChem. 2023 Oct 4;24(19):e202300467. doi: 10.1002/cbic.202300467

Guarrochena X, Kaudela B, Mindt TL. Automated solid-phase synthesis of metabolically stabilized triazolo-peptidomimetics. Journal of Peptide Science. 2023 Sept;29(9):e3488. doi: 10.1002/psc.3488

Wang Y, Staudinger JN , Mindt TL, Gasser G. Theranostics with photodynamic therapy for personalized medicine: to see and to treat. Theranostics. 2023;13(15):5501-5544. doi: 10.7150/thno.87363